Epigenetic proteins that place a histone mark.
servable in this model
measured here and in at least one other family
involving this family
| Quantity | Value |
|---|---|
| Measurements | 887 |
| Activity range, pActivity | 2.94 to 9.8 |
| Median activity | 5.76 |
| Endpoint | Measurements |
|---|---|
| IC50 | 827 |
| Ki | 44 |
| Kd | 15 |
| EC50 | 1 |
Every ligand counted here is measured in this family and in at least one other. The question worth asking is how many families a compound reaches altogether, because a compound seen in four families is a very different starting point from one seen in two.
| Families a compound reaches | Compounds |
|---|---|
| Two | 217 |
| Three | 21 |
| Four or more | 30 |
| Family | Shared compounds |
|---|---|
| Transferase | 96 |
| Eraser | 67 |
| Kinase | 35 |
| Oxidoreductase | 31 |
| Reader | 31 |
| Family A G protein-coupled receptor | 30 |